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Chemical Structure : EZH2-IN-3
Catalog No.: PC-62468Not For Human Use, Lab Use Only.
EZH2-IN-3 is a highly selective small molecule inhibitor of EZH2 and EZH1 with IC50 of 21/197/213 nM for wt EZH2/EZH2 Y641N/wt EZH1 respectively.
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EZH2-IN-3 is a highly selective small molecule inhibitor of EZH2 and EZH1 with IC50 of 21/197/213 nM for wt EZH2/EZH2 Y641N/wt EZH1 respectively; suppresses global histone H3-lysine 27 methylation and cause selective proliferation defects.
| M.Wt | 490.004 | |
| Formula | C27H28ClN5O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Garapaty-Rao S, et al. Chem Biol. 2013 Nov 21;20(11):1329-39.
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