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Fasitibant

Chemical Structure : Fasitibant

CAS No.: 869880-33-1

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Fasitibant (MEN16132, MEN-16132)

Catalog No.: PC-26631Not For Human Use, Lab Use Only.

Fasitibant (MEN16132) is a potent, selective, nonpeptide antagonist of type 2 bradykinin receptor (B2R) with pIC50 of 10.5 for [3H]-BK binding in mouse lung.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Fasitibant (MEN16132) is a potent, selective, nonpeptide antagonist of type 2 bradykinin receptor (B2R) with pIC50 of 10.5 for [3H]-BK binding in mouse lung.

Physicochemical Properties

M.Wt 836.69
Formula C36H50Cl4N6O6S
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(S)-4-amino-5-(4-(4-((2,4-dichloro-3-(((2,4-dimethylquinolin-8-yl)oxy)methyl)phenyl)sulfonamido)tetrahydro-2H-pyran-4-carbonyl)piperazin-1-yl)-N,N,N-trimethyl-5-oxopentan-1-aminium chloride hydrochloride

References

1. Valenti C, et al. Br J Pharmacol. 2012 Jun;166(4):1403-10.

2. Cialdai C, et al. J Pharmacol Exp Ther. 2009 Dec;331(3):1025-32.

3. Meini S, et al. Br J Pharmacol. 2007 Feb;150(3):313-20.

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