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Chemical Structure : GPR56 agonist 36
Catalog No.: PC-20909Not For Human Use, Lab Use Only.
GPR56 agonist 36 is a potent selective agonist of adhesion GPCR ADGRG1/GPR56 with EC50 of 2.95 uM.
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GPR56 agonist 36 is a potent selective agonist of adhesion GPCR ADGRG1/GPR56 with EC50 of 2.95 uM.
GPR56 agonist 36 activates GPR56 F385A/M389A and GPR56 L388A/M389A double TA mutant holoreceptors.
GPR56 agonist 36 shows exclusive specificity for GPR56 in a small panel of adhesion GPCRs and two class A GPCRs. ADGRG5/GPR114, ADGRG3/GPR97, and ADGRG1/GPR56 are from the same adhesion GPCR subfamily.
| M.Wt | 432.36 | |
| Formula | C22H26BrNO3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Alexander L Vizurraga, et al. Mol Pharmacol. 2023 Jun 8;MOLPHARM-AR-2023-000688.
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