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Chemical Structure : GSK 494581A
Catalog No.: PC-60676Not For Human Use, Lab Use Only.
GSK 494581A is a potent, specific and mixed glycine transporter subtype 1 (GlyT1) inhibitor (pIC50=7.7) and GPR55 agonist (pEC50=6.5).
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GSK 494581A is a potent, specific and mixed glycine transporter subtype 1 (GlyT1) inhibitor (pIC50=7.7) and GPR55 agonist (pEC50=6.5).
GSK 494581A shows no activity across a set of more than 200 validated molecular target assays from diverse classes, including kinases, proteases and other enzymes, GPCRs.
| M.Wt | 514.588 | |
| Formula | C27H28F2N2O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Brown AJ, et al. J Pharmacol Exp Ther. 2011 Apr;337(1):236-46.
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