JZ128 | PKN3 inhibitor | Probechem Biochemicals

Chemical Structure : JZ128

JZ128 (JZ-128)

Catalog No.: PC-26113Not For Human Use, Lab Use Only.

JZ128 is a selective, covalent inhibitor of Protein Kinase N3 (PKN3) with IC50 of 120 nM, targets Cys840 in PKN3, has no activity against CDK7 or CDK12/13.

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Biological Activity

JZ128 is a selective, covalent inhibitor of Protein Kinase N3 (PKN3) with IC50 of 120 nM, targets Cys840 in PKN3, has no activity against CDK7 or CDK12/13.

Physicochemical Properties

M.Wt	545.65
Formula	C32H31N7O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(E)-4-(4-(dimethylamino)but-2-enamido)-N-(3-((4-(4-methyl-1H-indol-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide

References

1. Browne CM, et al. J Am Chem Soc. 2019 Jan 9;141(1):191-203.

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JZ128 (JZ-128)

Biological Activity

Physicochemical Properties

References

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