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Chemical Structure : Ketanserin
CAS No.: 74050-98-9
Catalog No.: PC-42653Not For Human Use, Lab Use Only.
A high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 100 mg | $56 | In stock | |
| 1 g | Get quote |
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A high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C; also has a high affinity antagonist for the H1 receptor (Ki= 2 nM) and α1-adrenergic receptor (Ki=40 nM); an antihypertensive agent.
Hypertension
Approved
| M.Wt | 395.4268 | |
| Formula | C22H22FN3O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: 8 mg/mL |
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| Chemical Name/SMILES |
2,4(1H,3H)-Quinazolinedione, 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]- |
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1. Creed-Carson M, et al. Behav Brain Res. 2011 Jun 1;219(2):273-9.
2. Catafau AM, et al. J Cereb Blood Flow Metab. 2010 May;30(5):985-93.
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