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Chemical Structure : ML250
CAS No.: 1421365-63-0
Catalog No.: PC-38611Not For Human Use, Lab Use Only.
ML250 (CYM 50769) is a potent and selective GPR7 (Neuropeptides B/W receptor 1, NPBWR1) antagonist probe, inhibits human GPR7 expression in the presence of GPR7 agonist NPW with IC50 value of 124 nM-244 nM, displays 82- >161 fold selectivity over MCH1.
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|---|---|---|---|
| 10 mg | $158 | In stock | |
| 25 mg | $278 | In stock | |
| 50 mg | $488 | In stock | |
| 100 mg | Get quote |
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ML250 (CYM 50769) is a potent and selective GPR7 (Neuropeptides B/W receptor 1, NPBWR1) antagonist probe, inhibits human GPR7 expression in the presence of GPR7 agonist NPW with IC50 value of 124 nM-244 nM, displays 82- >161 fold selectivity over MCH1.
| M.Wt | 416.861 | |
| Formula | C24H17ClN2O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
5-chloro-2-(9H-fluoren-9-yl)-4-(4-methoxyphenoxy)pyridazin-3(2H)-one |
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1. Miguel Guerrero, et al. In: Probe Reports from the NIH Molecular Libraries Program [Internet].
2. Miguel Guerrero, et al. Bioorg Med Chem Lett. 2013 Feb 1;23(3):614-9.
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