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Chemical Structure : PFI-4
CAS No.: 900305-37-5
Catalog No.: PC-45507Not For Human Use, Lab Use Only.
PFI-4 is a potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.3.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $88 | In stock | |
| 25 mg | $138 | In stock | |
| 50 mg | $218 | In stock | |
| 100 mg | Get quote |
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PFI-4 is a potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.3.
PFI-4 exhibits >100-fold selectivity for BRPF1 over a panel of other bromodomains including BRPF2 (BRD1), BRPF3 and BRD4.
| M.Wt | 380.4402 | |
| Formula | C21H24N4O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: 26 mg/mL |
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| Chemical Name/SMILES |
Benzamide, N-[2,3-dihydro-1,3-dimethyl-2-oxo-6-(1-pyrrolidinyl)-1H-benzimidazol-5-yl]-2-methoxy- |
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1. Demont EH, et al. ACS Med Chem Lett. 2014 Sep 10;5(11):1190-5.
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