Photoazolol-1 (PZL-1)

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Chemical Structure : Photoazolol-1

Catalog No.: PC-28009Not For Human Use, Lab Use Only.

Photoazolol-1 is a photoswitchable β2-adrenergic receptor (β2AR) blocker (β-blocker) with pEC50 of 7.73 (Dark, trans-photoazolol-1), 52-fold selective over under light condition (cis-photoazolol-1, pEC50=6.01).

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Photoazolol-1 is a photoswitchable β2-adrenergic receptor (β2AR) blocker (β-blocker) with pEC50 of 7.73 (Dark, trans-photoazolol-1), 52-fold selective over under light condition (cis-photoazolol-1, pEC50=6.01).

Physicochemical Properties

M.Wt	370.45
Formula	C20H26N4O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-N-(4-((2-(2-hydroxy-3-(isopropylamino)propoxy)phenyl)diazenyl)phenyl)acetamide

References

1. Stipp R, et al. Angew Chem Int Ed Engl. 2026 Apr 27;65(18):e17995.

2. Anna Duran-Corbera, et al. J Med Chem. 2020 Aug 13;63(15):8458-8470.

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