Pimecrolimus | Calcineurin inhibitor | Probechem Biochemicals

Chemical Structure : Pimecrolimus

CAS No.: 137071-32-0

Catalog No.: PC-26136Not For Human Use, Lab Use Only.

Pimecrolimus (SDZ-ASM 981) is a potent, nonsteroid and orally active calcineurin inhibitor with Ki of 117 nM, shows anti-inflammatory activity.

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25 mg	$58	In stock
100 mg	$98	In stock
250 mg	$148	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Pimecrolimus (SDZ-ASM 981) is a potent, nonsteroid and orally active calcineurin inhibitor with Ki of 117 nM, shows anti-inflammatory activity.

M.Wt	810.46
Formula	C43H68ClNO11
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(3S,4R,5S,8R,9E,12S,14S,15R,16S,18R,19R,26aS)-3-[(1E)-2-[(1R,3R,4S)-4-Chloro-3-methoxycyclohexyl]-1-methylethenyl]-8-ethyl-5,6,8,11,12,13,14,15,16,17,18,19,24,25,26,26a-hexadecahydro-5,19-dihydroxy-14,16-dimethoxy-4,10,12,18-tetramethyl-15,19-epoxy-3H-pyr

1. Grassberger M, et al. Br J Dermatol. 1999 Aug;141(2):264-73.

2. Bochelen D, et al. J Pharmacol Exp Ther. 1999 Feb;288(2):653-9.