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Chemical Structure : Pitolisant hydrochloride
CAS No.: 903576-44-3
Catalog No.: PC-42911Not For Human Use, Lab Use Only.
A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 50 mg | $384 | In stock |
Bulk size, bulk discount!
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A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM; no effect on H1, H2, H4 receptors (IC50>10 uM); orally bioactive.
Sleep Disorder
Approved
| M.Wt | 332.3084 | |
| Formula | C17H27Cl2NO | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 43 mg/mL |
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| Chemical Name/SMILES |
Piperidine, 1-[3-[3-(4-chlorophenyl)propoxy]propyl]-, hydrochloride (1:1) |
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1. Ligneau X, et al. J Pharmacol Exp Ther. 2007 Jan;320(1):365-75.
2. Dudek M, et al. Metab Brain Dis. 2016 Oct;31(5):1023-9.
3. Ligneau X, et al. Biochem Pharmacol. 2007 Apr 15;73(8):1215-24.
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