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SR-49059

Chemical Structure : SR-49059

CAS No.: 150375-75-0

SR-49059 (SR49059)

Catalog No.: PC-21436Not For Human Use, Lab Use Only.

SR49059 (SR-49059) is a potent, selective and orally active vasopressin V1a antagonist with Ki of 1.4 nM.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

SR49059 (SR-49059) is a potent, selective and orally active vasopressin V1a antagonist with Ki of 1.4 nM.

Physicochemical Properties

M.Wt 620.50
Formula C28H27Cl2N3O7S
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

(2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4-diMethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxaMide

References

1. Méchaly I, et al. Eur J Pharmacol. 1999 Nov 3;383(3):287-90.

2. Tahara A, et al. Br J Pharmacol. 1998 Dec;125(7):1463-70.

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