| Cat. No. |
Product Name |
Information |
| PC-36095 |
Pecavaptan
V1a/V2 receptor antagonist
|
Pecavaptan (BAY 1753011) is a potent, orally active and dual antagonist of vasopressin receptor V1a/V2 receptor (Ki=0.5 nM and 0.6 nM for human, respectively). |
| PC-70166 |
Conivaptan
Vasopressin Receptor inhibitor
|
Conivaptan (YM-087) is a potent, selective, nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively. |
| PC-60078 |
RG7713
V1a receptor antagonist
|
RG7713 (RO5028442, RG-7713) is a potent, highly selective, brain-penetrant vasopressin 1a (hV1a) antagonist with Ki of 1 nM. |
| PC-60033 |
Balovaptan
V1a receptor antagonist
|
Balovaptan (RG7314, RO5285119) is a potent, selective vasopressin-1 receptor antagonist with Kb of 0.39 nM at the human V1a receptor. |
| PC-47487 |
Ornipressin
|
Ornipressin is a vasoconstrictor, haemostatic and renal agent. |
| PC-45192 |
Desmopressin
|
Desmopressin is a synthetic analogue of the antidiuretic hormone arginine vasopressin. |
| PC-45191 |
Desmopressin acetate
|
Desmopressin acetate is a synthetic analogue of the antidiuretic hormone arginine vasopressin. |
| PC-45459 |
Mozavaptan
|
Mozavaptan (OPC-31260) is a potent, selective nonpeptide vasopressin V2 receptor antagonist with IC50 of 14 nM. |
| PC-45460 |
Conivaptan hydrochloride
Vasopressin Receptor inhibitor
|
Conivaptan (YM-087) is a potent, selective nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively. |
| PC-45125 |
Tolvaptan
V2 antagonist
|
Tolvaptan (OPC-41061) is a highly potent selective, competitive vasopressin V2-receptor antagonist with Ki of 0.43 nM, >200-fold more selective than for V1A-receptors. |
| PC-21617 |
PF-184563
V1a receptor antagonist
|
PF-184563 is a potent and selective vasopressin V1a antagonist with IC50 of 6.7 nM (hV1a). |
| PC-21616 |
Relcovaptan
V1a receptor antagonist
|
SR 49059 (SR-49059) is a potent, selective and orally active vasopressin V1a antagonist with Ki of 1.4 nM. |
