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Chemical Structure : Sarpogrelate hydrochloride
CAS No.: 135159-51-2
Catalog No.: PC-42655Not For Human Use, Lab Use Only.
A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 50 mg | $188 | In stock | |
| 100 mg | $256 | In stock |
Bulk size, bulk discount!
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A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B; displays selectivity over 5-HT1-like, 5-HT3, beta, H1, H2 and M3; blocks serotonin-induced platelet aggregation.
Heart Failure
Approved
| M.Wt | 465.967 | |
| Formula | C24H32ClNO6 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 62 mg/mL |
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| Chemical Name/SMILES |
Butanedioic acid, 1-[2-(dimethylamino)-1-[[2-[2-(3-methoxyphenyl)ethyl]phenoxy]methyl]ethyl] ester, hydrochloride (1:1) |
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1. Kikumoto R, et al. J Med Chem. 1990 Jun;33(6):1818-23.
2. Pertz H, et al. J Pharm Pharmacol. 1995 Apr;47(4):310-6.
3. Nishio H, et al. Arch Int Pharmacodyn Ther. 1996 Mar-Apr;331(2):189-202.
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