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T-10418

Chemical Structure : T-10418

CAS No.: 1608784-68-4

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T-10418 (T10418)

Catalog No.: PC-22564Not For Human Use, Lab Use Only.

T-10418 is a potent, selective agonist of G protein-coupled receptor G2A (GPR132) with EC50 of 0.82 uM.

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10 mg $398 In stock
25 mg $598 In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

T-10418 is a potent, selective agonist of G protein-coupled receptor G2A (GPR132) with EC50 of 0.82 uM.
T-10418 exhibits higher potency than the reference and natural ligand 9-HODE and high selectivity among G protein-coupled receptors.
T-10418 has favorable activity, a clean selectivity profile, excellent solubility, and high metabolic stability, is a pharmacological tool to investigate the effects of G2A activation.

Physicochemical Properties

M.Wt 376.41
Formula C22H20N2O4
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
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Solubility

10 mM in DMSO
Chemical Name/SMILES

(3-(pyridin-3-ylmethoxy)benzoyl)-D-phenylalanine

References

1. Hernandez-Olmos V, et al. J Med Chem. 2024 Jun 25. doi: 10.1021/acs.jmedchem.3c02164.

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