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Chemical Structure : TPCA-1
CAS No.: 507475-17-4
Catalog No.: PC-42243Not For Human Use, Lab Use Only.
TPCA-1 (IKK-2 Inhibitor IV) is a potent, selective and orally bioavailable IKK-2 inhibitor with IC50 of 63 nM, TNF cell IC50 of 0.4 uM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $88 | In stock | |
| 25 mg | $138 | In stock | |
| 50 mg | $218 | In stock | |
| 100 mg | Get quote |
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TPCA-1 (IKK-2 Inhibitor IV) is a potent, selective and orally bioavailable IKK-2 inhibitor with IC50 of 63 nM, TNF cell IC50 of 0.4 uM.
TPCA-1 displays >100-fold selectivity over IKK-1.
| M.Wt | 279.2901 | |
| Formula | C12H10FN3O2S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
3-Thiophenecarboxamide, 2-[(aminocarbonyl)amino]-5-(4-fluorophenyl)- |
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1. Baxter A, et al. Bioorg Med Chem Lett. 2004 Jun 7;14(11):2817-22.
2. Park BK, et al. Nat Med. 2007 Jan;13(1):62-9.
3. Amaya M, et al. PLoS One. 2014 Feb 19;9(2):e86745.
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