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Chemical Structure : TRPV2 antagonist SET2
CAS No.: 2313525-20-9
Catalog No.: PC-22170Not For Human Use, Lab Use Only.
SET2 is a potent, subtype-selective inhibitor of transient receptor potential vanilloid type 2 (TRPV2) with IC50 of 0.46 uM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $98 | In stock | |
| 10 mg | $148 | In stock | |
| 25 mg | $258 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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SET2 is a potent, subtype-selective inhibitor of transient receptor potential vanilloid type 2 (TRPV2) with IC50 of 0.46 uM.
SET2 displays no activity against TRPV1, TRPV3, or TRPV4.
SET2 (0-20 uM) inhibits the migration of prostate cancer cell PC-3M expressing TRPV2.
| M.Wt | 402.44 | |
| Formula | C17H21F3N4O2S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
N-(Furan-2-ylmethyl)-3-((4-(methyl(propyl)amino)-6-(trifluoromethyl)pyrimidin-2-yl)thio)propanamide |
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1. Hao Chai, et al. J Med Chem. 2019 Feb 14;62(3):1373-1384.
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