Welcome to Shanghai Probechem Biochemicals Co Ltd !Global Supplier of Chemical Probes, Inhibitors & Agonists.
Chemical Structure : Tenalisib
CAS No.: 1639417-53-0
Catalog No.: PC-60567Not For Human Use, Lab Use Only.
Tenalisib (RP-6530) is a potent, selective, orally active p110δ/γ PI3K dual inhibitor with IC50 of 24.5 and 33.2 nM, respectively.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $128 | In stock | |
| 25 mg | $218 | In stock | |
| 50 mg | $378 | In stock | |
| 100 mg | Get quote |
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
Tenalisib (RP-6530) is a potent, selective, orally active p110δ/γ PI3K dual inhibitor with IC50 of 24.5 and 33.2 nM, respectively.
Tenalisib (RP-6530) displays good selectivity over p110α (>300-fold) and p110β (>100-fold) isoforms.
Tenalisib (RP-6530) inhibits LPS induced CD19+ cell proliferation in human whole blood with EC50 of 250 nM, and LPS induced CD45R+ cell proliferation in mouse whole blood with EC50 of 101 nM.
Tenalisib (RP-6530) shows the potential for treatment of cancer and inflammation diseases.
| M.Wt | 415.43 | |
| Formula | C23H18FN5O2 | |
| Appearance | Solid | |
| Storage |
|
|
| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
(S)-2-(1-((7H-purin-6-yl)amino)propyl)-3-(3-fluorophenyl)-4H-chromen-4-one |
|
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright
