Tilpisertib fosmecarbil (GS-5290) | TPL2 inhibitor

Chemical Structure : Tilpisertib fosmecarbil

Tilpisertib fosmecarbil (GS-5290, GS5290)

Catalog No.: PC-27855Not For Human Use, Lab Use Only.

Tilpisertib fosmecarbil (GS-5290) is an intestinally cleaved prodrug of GS-4875, a potent tumor progression locus 2 (TPL2 , COT, MAP3K8) inhibitor.

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Biological Activity

Tilpisertib fosmecarbil (GS-5290) is an intestinally cleaved prodrug of GS-4875, a potent tumor progression locus 2 (TPL2 , COT, MAP3K8) inhibitor.

Physicochemical Properties

M.Wt	747.15
Formula	C35H36ClN8O7P
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(phosphonooxy)methyl (S)-((1-(bicyclo[1.1.1]pentan-1-yl)-1H-1,2,3-triazol-4-yl)(2-methyl-1-oxo-1,2-dihydroisoquinolin-5-yl)methyl)(8-chloro-3-cyano-4-(neopentylamino)quinolin-6-yl)carbamate

References

1. Priyanka A Madia, et al. J Clin Pharmacol. 2026 Aug;66(8):e70269.

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Tilpisertib fosmecarbil (GS-5290, GS5290)

Biological Activity

Physicochemical Properties

References

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