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Chemical Structure : UCPH-102
Catalog No.: PC-62149Not For Human Use, Lab Use Only.
UCPH-102 is a selective, brain penetrant inhibitor of EAAT1 (Excitatory amino acid transporter 1) with IC50 of 420 nM.
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UCPH-102 is a selective, brain penetrant inhibitor of EAAT1 (Excitatory amino acid transporter 1) with IC50 of 420 nM; exhibits no inhibitory activity aganist EAAT2-5 (>300 uM); has been shown to cross the blood-brain barrier, and become a valuable tool for studying the role of EAAT1 in brain.
| M.Wt | 330.387 | |
| Formula | C21H18N2O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Huynh TH, et al. Bioorg Med Chem. 2012 Dec 1;20(23):6831-9.
2. Haym I, et al. ChemMedChem. 2016 Feb 17;11(4):403-19.
3. Erichsen MN, et al. Neurochem Res. 2014 Oct;39(10):1964-79.
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