Welcome to Shanghai Probechem Biochemicals Co Ltd !Global Supplier of Chemical Probes, Inhibitors & Agonists.
Chemical Structure : VU6047534
Catalog No.: PC-21829Not For Human Use, Lab Use Only.
VU6047534 is a selective, peripherally restricted 5-HT2B partial agonist with IC50 of 480 nM in radioligand binding assays.
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
VU6047534 is a selective, peripherally restricted 5-HT2B partial agonist with IC50 of 480 nM in radioligand binding assays.
VU6047534 shows high subtype selectivity relative to 5-HT2A and 5-HT2C (no significant inhibition up to 10 uM).
VU6047534 is peripherally restricted and able to both prevent and treat Sugen-hypoxia-induced pulmonary arterial hypertension.
| M.Wt | 351.42 | |
| Formula | C19H17N3O2S | |
| Appearance | Solid | |
| Storage |
|
|
| Solubility |
10 mM in DMSO |
|
1. Valentine MS, et al.JACC Basic Transl Sci. 2023 Sep 13;8(10):1379-1388.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright
