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Chemical Structure : Varlitinib
CAS No.: 845272-21-1
Catalog No.: PC-42640Not For Human Use, Lab Use Only.
Varlitinib (ARRY-334543) is a potent, orally active, ATP-competitive, selective, reversible inhibitor of ErbB1 and ErbB2.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $152 | In stock | |
| 50 mg | $432 | In stock | |
| 100 mg | $592 | In stock | |
| 1 g | Get quote |
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Varlitinib (ARRY-334543) is a potent, orally active, ATP-competitive, selective, reversible inhibitor of ErbB1 and ErbB2; significantly reverses ABCG2-MDR by directly inhibiting the drug efflux function of ABCG2 at 1.0 uM; significantly reverses drug resistance mediated by ABCG2.
Thyroid Cancer
Approved
| M.Wt | 466.9433 | |
| Formula | C22H19ClN6O2S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: 16.67 mg/mL |
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| Chemical Name/SMILES |
4,6-Quinazolinediamine, N4-[3-chloro-4-(2-thiazolylmethoxy)phenyl]-N6-[(4R)-4,5-dihydro-4-methyl-2-oxazolyl]- |
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1. Wang DS, et al. J Cell Biochem. 2014 Aug;115(8):1381-91.
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