You are here:Home-Chemical Inhibitors & Agonists-Epigenetics-Histone Methyltransferase (HMTase)-WDR5-0103
WDR5-0103

Chemical Structure : WDR5-0103

CAS No.: 890190-22-4

WDR5-0103 (WD-Repeat Protein 5-0103)

Catalog No.: PC-45617Not For Human Use, Lab Use Only.

A potent MLL1-WDR5 interaction inhibitor with IC50 of 26.4 nM in competitive binding assay.

Packing Price Stock Quantity
10 mg $80 In stock
50 mg $320 In stock
100 mg $520 In stock

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

A potent MLL1-WDR5 interaction inhibitor with IC50 of 26.4 nM in competitive binding assay; inhibits the catalytic activity of MLL1 complex with IC50 value of 5.4 uM.

Physicochemical Properties

M.Wt 383.4409
Formula C21H25N3O4
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

DMSO: ≥ 40 mg/mL

Chemical Name/SMILES

Benzoic acid, 3-[(3-methoxybenzoyl)amino]-4-(4-methyl-1-piperazinyl)-, methyl ester

References

1. Li DD, et al. Bioorg Med Chem. 2016 Nov 15;24(22):6109-6118.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: