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Chemical Structure : YEATS4 binder 4e
Catalog No.: PC-49599Not For Human Use, Lab Use Only.
YEATS4 binder 4e is a potent, selective small-molecule epigenetic reader YEATS4 binder with Ki of 37 nM, >15-fold selectivity over YEATS1, 2 and 3.
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YEATS4 binder 4e is a potent, selective small-molecule epigenetic reader YEATS4 binder with Ki of 37 nM, >15-fold selectivity over YEATS1, 2 and 3.
YEATS4 binder 4e directly binds to YEATS4 at the lysine acetylation recognition site of the YEATS domain.
YEATS4 binder 4e engages YEATS4 with nanomolar potency in a whole-cell nanoluciferase bioluminescent resonance energy transfer assay (IC50=300 nM).
| M.Wt | 414.55 | |
| Formula | C23H34N4O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Allyn T Londregan, et al. J Med Chem. 2022 Dec 23. doi: 10.1021/acs.jmedchem.2c01421.
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