Cat. No. |
Product Name |
Information |
PC-61052 |
hTG2 inhibitor VA4
hTG2 inhibitor
|
hTG2 inhibitor VA4(VA4) is a novel potent, irreversible inhibitor of human tissue transglutaminase (hTG2) with Ki of 12.9 uM, allosterically abolishs its GTP binding ability with a high degree of selectivity and efficiency. |
PC-45039 |
LDN-27219
TGase inhibitor
|
LDN-27219 is a potent, reversible inhibitor of hTGase (Tissue transglutaminase) with IC50 of 0.8 uM. |
PC-24404 |
TG2 inhibitor 1-155
TG2 inhibitor
|
TG2 inhibitor 1-155 (TG2 inhibitor 3h) is a potent, selective small molecule Transglutaminase 2 (TG2, TGase2, TGM2) inhibitor with IC50 of 6.1 nM, >1000-fold selective over TG1, TG3, TG6, and Factor XIIIa (FXIIIa). |
PC-21821 |
IPN60090
GLS-1 inhibitor
|
IPN60090 (IACS-6274) is a potent, selective glutaminase-1 (GLS-1) inhibitor with IC50 of 31 nM, inhibits proliferation of A549 cells with IC50 of 26 nM. |