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Chemical Structure : AM-630
CAS No.: 164178-33-0
Catalog No.: PC-60760Not For Human Use, Lab Use Only.
AM-630 (6-Iodopravodoline) is a potent and selective inverse agonist for the cannabinoid receptor CB2 with Ki of 32.1 nM, 165-fold selectivity over CB1.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 25 mg | $198 | In stock | |
| 100 mg | $498 | In stock | |
| 200 mg | Get quote | ||
| 1 g | Get quote |
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AM-630 (6-Iodopravodoline) is a potent and selective inverse agonist for the cannabinoid receptor CB2 with Ki of 32.1 nM, 165-fold selectivity over CB1.
AM-630 inhibits forskolin-stimulated cyclic AMP production in CB1-transfected cells (22.6% at 1 uM and 45.9% at 10 uM).
| M.Wt | 504.4 | |
| Formula | C23H25IN2O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
[6-iodo-2-methyl-1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl](4-methoxyphenyl)-methanone |
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1. Ross RA, et al. Br J Pharmacol. 1999 Feb;126(3):665-72.
2. Malan TP Jr, et al. Pain. 2001 Sep;93(3):239-45.
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