Chemical Structure : Cligosiban
Catalog No.: PC-61369Not For Human Use, Lab Use Only.
A potent, specific oxytocin receptor antagonist with Ki of 9.5 nM, displays high selectivity over the vasopressin receptors.
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A potent, specific oxytocin receptor antagonist with Ki of 9.5 nM, displays high selectivity over the vasopressin receptors; demonstrates excellent potency and selectivity, as well as promising in vivo pharmacokinetics and significantly improved aqueous solubility.
Sexual Dysfunction
Phase 1 Discontinued
M.Wt | 419.841 | |
Formula | C19H19ClFN5O3 | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
1. Vidal B, et al. Nucl Med Biol. 2017 Dec;55:1-6.
2. Brown A, et al. Bioorg Med Chem Lett. 2010 Jan 15;20(2):516-20.
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