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Chemical Structure : GSK-1842799
Catalog No.: PC-61604Not For Human Use, Lab Use Only.
GSK-1842799 is a potent, selective, oral bioavailable S1P1 agonist with bind affinity of 0.52 nM.
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GSK-1842799 is a potent, selective, oral bioavailable S1P1 agonist with bind affinity of 0.52 nM.
GSK-1842799 displays an excellent selectivity (>3,000-fold) for S1P1 over S1P3.
GSK-1842799 significantly reduces blood lymphocyte at 3 mg/kg, achieves efficacy equivalent to FTY720 in the mouse EAE model of MS.
| M.Wt | 431.518 | |
| Formula | C20H28F3N3O2S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Deng H, et al. ACS Med Chem Lett. 2013 Aug 27;4(10):942-7.
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