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Chemical Structure : GSK-2239633
Catalog No.: PC-61980Not For Human Use, Lab Use Only.
GSK-2239633 is a potent, selective, allosteric CCR4 antagonist with pIC50 of 7.96.
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GSK-2239633 is a potent, selective, allosteric CCR4 antagonist with pIC50 of 7.96; also inhibits TARC-induced increases in the F-actin content of isolated human CD4+ CCR4+ T-cells with pA2 of 7.1.
Asthma
Phase 1 Clinical
| M.Wt | 506.976 | |
| Formula | C21H19ClN4O5S2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Cahn A, et al. BMC Pharmacol Toxicol. 2013 Feb 28;14:14.
2. Procopiou PA, et al. Bioorg Med Chem Lett. 2012 Apr 15;22(8):2730-3.
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