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Chemical Structure : GSK-864
CAS No.: 1816331-66-4
Catalog No.: PC-45645Not For Human Use, Lab Use Only.
GSK-864 is a compound structurally related to GSK321 with improved in vivo pharmacokinetic properties.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $178 | In stock | |
| 25 mg | $328 | In stock | |
| 50 mg | $528 | In stock | |
| 100 mg | Get quote |
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GSK-864 is a compound structurally related to GSK321 with improved in vivo pharmacokinetic properties.
GSK-864 shows the similar activity (2-HG production in R132C IDH1 mutant HT1080 fibrosarcoma cells, EC50 of 320 nM).
GSK-864 reduces leukemic blasts in vivo.
| M.Wt | 558.6033 | |
| Formula | C30H31FN6O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 100 mg/mL |
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| Chemical Name/SMILES |
(S)-1-(4-fluorobenzyl)-N3-(4-methoxy-3,5-dimethylphenyl)-7-methyl-5-(1H-pyrrole-2-carbonyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine-3,7-dicarboxamide |
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1. Okoye-Okafor UC, et al. Nat Chem Biol. 2015 Nov;11(11):878-86.
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