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Chemical Structure : LPA2-IN-1
CAS No.: 1017606-66-4
Catalog No.: PC-45411Not For Human Use, Lab Use Only.
A potent, selective LPA2 (EDG4) antagonist with IC50 of 17 nM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $400 | In stock | |
| 50 mg | $1200 | In stock | |
| 100 mg | $1680 | In stock |
Bulk size, bulk discount!
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A potent, selective LPA2 (EDG4) antagonist with IC50 of 17 nM; inhibits the phosphorylation of Erk induced by LPA in a concentration dependent manner; inhibits HCT-116 colon cancer cell proliferation caused by LPA in a doses dependent manner.
| M.Wt | 500.4649 | |
| Formula | C20H23Cl2N5O2S2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
Thieno[3,2-d]pyrimidin-4-amine, N-[(1S)-2-[4-[(3,4-dichlorophenyl)sulfonyl]-1-piperazinyl]-1-methylethyl]-7-methyl- |
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1. Beck HP, et al. Bioorg Med Chem Lett. 2008 Feb 1;18(3):1037-41.
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