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Chemical Structure : SAR-216471 hydrochloride
Catalog No.: PC-61535Not For Human Use, Lab Use Only.
SAR-216471 is a potent, highly selective, intravenous and oral, reversible P2Y12 receptor antagonist with binding IC50 of 17 nM.
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SAR-216471 is a potent, highly selective, intravenous and oral, reversible P2Y12 receptor antagonist with binding IC50 of 17 nM; inhibits ADP-induced platelet aggregation in human platelet rich plasma with IC50 of 0.1 uM; exhibits an ED50 of 2.75mg/kg in ex vivo platelet aggregation model in rats.
| M.Wt | 599.51 | |
| Formula | C28H31ClN8O3.HCl | |
| Appearance | Solid | |
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| Solubility |
10 mM in DMSO |
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1. Boldron C, et al. J Med Chem. 2014 Sep 11;57(17):7293-316.
2. Delesque-Touchard N, et al. Thromb Res. 2014 Sep;134(3):693-703.
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