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Request The Product List ofBombesin Receptor Bombesin Receptor

Cat. No. Product Name CAS No. Information
PC-61219

RC-3095

138147-78-1 A potent, peptide bombesin/gastrin releasing peptide (GRPR,BRS-1) antagonist.

Solid Tumors

Phase 2 Discontinued

PC-61218

BRS-3 agonist Compound A racemate

A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 270/130 nM for human/rat BRS-3, respectively; displays no activity against GRPR (BRS-1) and NMBR (BRS-2) (EC50>10 uM).
PC-61217

(S)-BRS-3 agonist Compound A

The distomer of BRS-3 agonist Compound A, shows no activity for bombesin receptor subtype-3 (BRS-3) with EC50>10 uM.
PC-61216

BRS-3 agonist Compound A

A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 250/100 nM for human/rat BRS-3, resp+H1437+M1438
PC-61215

Bantag-1 trifluoroacetate

A potent, highly selective, peptide bombesin receptor subtype-3 (BRS-3) antagonist with IC50 of 2-8 nM for human and rodent BRS-3, displays 1000-fold selectivity over hNMBR and hGRPR, increases food intake and produces an obesity phenotype in mice.

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