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Cat. No. Product Name Information
PC-20049

PF-04457845

FAAH inhibitor

PF-04457845 (Redafamdastat) is a highly potent, selective and covalent fatty acid amide hydrolase (FAAH) inhibitor with IC50 of 7.2 nM (human FAAH).
PC-49841

UCM1341

FAAH inhibitor

UCM1341 (UCM 1341) is a bivalent ligand with melatonin receptor agonist (hMT1/hMT2, pKi=9.11/8.77) and fatty acid amide hydrolase (FAAH) inhibitory activity (rFAAH IC5=0.85 nM).
PC-49009

PF-3845

FAAH inhibitor

PF-3845 is a potent, highly selective, covalent FAAH inhibitor with Ki of 0.23 uM, highly selective for FAAH in the brain.
PC-47021

ARN15381

FAAH inhibitor/D3 agonist

ARN15381 is a potent, multitarget FAAH inhibitor/D3 partial agonist with low nanomolar range activity, decreases nicotine self-administration in male rats.
PC-38511

ARN272

FLAT inhibitor

ARN272 (ARN-272) is a specific, competitive FAAH-like anandamide transporter (FLAT) inhibitor, antagonizes [3H]-anandamide binding to purified FLAT (IC50=1.8 uM) and inhibits [3H]-anandamide accumulation in FLAT-expressing HEK293 cells with IC50 of 3 uM.
PC-72178

PKM-833

FAAH inhibitor

PKM-833 (PKM833) is a potent, selective, and orally active FAAH inhibitor with IC50 of 8.8 and 10 nM against human and rat FAAH, respectively.
PC-38094

URB937

FAAH inhibitor

URB937 (URB 937) is a potent, peripherally restricted FAAH inhibitor with IC50 of 26.8 nM.
PC-63423

JNJ-40413269

FAAH inhibitor

JNJ-40413269 is a potent, selective, blood brain barrier (BBB) penetrant FAAH inhibitor with IC50 of 5.3 and 6.3 nM for hFAAH and rFAAH, respectively.
PC-63017

LY2318912

Anandamide transporter inhibitor

LY2318912 is a potent, competitive, small molecule inhibitor of anandamide uptake with IC50 of 7.27 nM, shows high affinity against anandamide transporter binding site with Kd of 7.62 nM.
PC-62533

SSR411298

FAAH inhibitor

SSR411298 is a highly selective, brain penetrant and orally-active inhibitor of FAAH with IC50 of 62.5 nM (mouse brain FAAH).
PC-60985

ASP 8477

FAAH inhibitor

ASP8477 is a novel potent, highly selective fatty acid amide hydrolase (FAAH) inhibitor with IC50 of 0.99, 1.65 and 57.3 nM for human FAAH-1, FAAH-1 (P129T) and FAAH-2, respectively.
PC-60706

SA57

FAAH/MAGL inhibitor

SA57a is a highly potent and selective dual FAAH/MAGL inhibitor with IC50 of 1-3 nM against FAAH, inhibits mouse (IC50=410 nM) and human (IC50=1.4 uM) MAGL.

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