| Cat. No. |
Product Name |
Information |
| PC-38251 |
TM-N1324
GPR39 agonist
|
GPR39 agonist Cpd1324 (TM-N1324) is a potent, selective, orally active GPR39 agonist, activats human GPR39 with high efficacy and potencies of 280 nM and 9 nM in the absence and presence of Zn2+, respectively. |
| PC-62255 |
GPR39 modulator 3
GPR39 modulator
|
GPR39 modulator 3 is a Hedgehog pathway inhibitor that has high cellular potency (EC50=5 nM) in the reporter gene assay, activates the orphan receptor GPR39 and potently reduces of Gli1 and Ptch1 mRNA levels. |
| PC-60593 |
TC G-1008
GPR39 agonist
|
TC G-1008 is a potent, selective, orally bioavailable GPR39 agonist with EC50 of 0.4 and 0.8 nM for rat and human GPR39, respectively. |
| PC-62256 |
GPR39 modulator 7
|
GPR39 modulator 7 is a Hedgehog pathway inhibitor that has high cellular potency (EC50=20 nM) in the reporter gene assay, activates the orphan receptor GPR39 and potently reduces of Gli1 and Ptch1 mRNA levels. |
