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Cat. No. Product Name Information
PC-49427

RXFP2 agonist 6641

FXRP2 agonist

RXFP2 agonist 6641 is a highly potent, selective and full allosteric agonist of relaxin/insulin-like family peptide receptor 2 (RXFP2) with EC50 of 0.38 uM, Emax=107% (hFXRP2).
PC-49353

AZD5462

RXFP1 agonist

AZD5462 (AZD-5462) is a selective, allosteric, oral agonist of the Relaxin family peptide receptor 1 (RXFP1) with pEC50 of 7.8 (hRXFP1).
PC-38726

RLX-33

RXFP3 antagonist

RLX-33 is a selective small-molecule nonpeptide antagonist of neuropeptide relaxin-3/RXFP3 with IC50 of 2.36 uM (cAMP functional assays), selective for RXFP3 over RXFP1 and RXFP4.
PC-70187

ML-290

RXFP1 agonist

ML-290 (ML290) is a potent and selective small-molecule agonist of hRXFP1 with EC50 of 94 nM.
PC-22033

AZ7976

RXFP1 agonist

AZ7976 (AZ-7976) is a potent, highly selective, allosteric relaxin family peptide receptor 1 (RXFP1) agonist with pEC50 of 9.4 in hRXFP1 cAMP assay in CHO-K1 cells, Emax=114%.
PC-20022

DC591053

RXFP4 agonist

DC591053 (DC 591053) is a selective small molecule agonist of relaxin family peptide receptor 4 (RXFP4) with pEC50  of 7.24  and pKi  of  6.95, shows no activity against RXFP3.
PC-49433

RXFP3/4 agonist 4

RXFP3/4 agonist

RXFP3/4 agonist 4 is a potent, selective, nonpeptide dual RXFP3/4 agonist with EC50 of 82/2.0 nM in cellualr cAMP assays.
PC-49432

RXFP3 agonist 10d

RXFP3/4 agonist

RXFP3 agonist 10d is a potent, selective, nonpeptide dual RXFP3/4 agonist with EC50 of 3.1/2.7 nM, no agonist activity against RXFP1 at 10 uM.

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