SB699551 is a potent, selective 5-HT5A receptor antagonist with pKi of 8.3, >100-fold sele..
FHD-286 (FHD286) is a highly potent, selective, allosteric and orally available inhibitor ..
BMS-986242 (BMS986242) is a potent, selective IDO1 inhibitor with IC50 of 2 nM in cellular..
MRTX-1133 (MRTX1133) is a potent, selective and noncovalent inhibitor KRAS G12D with SPR K..
CSRM617 (CSRM-617) is a small-molecule inhibitor of the transcription factor ONECUT2 (OC2)..
STING agonist diABZI compound 3 is an amidobenzimidazole (ABZI)-based compound that functi..
Exicorilant (CORT125281, CORT-125281) is a potent, selective glucocorticoid receptor (GR) ..
A potent, selective S1P3 antagonist with Ki of 0.25 nM; displays selectivity over other S1..
A potent, selective S1P3 antagonist with Ki of 0.25 nM; displays selectivity over other S1..
A novel potent, selective PDE5 inhibitor with IC50 of 0.056 nM for PDE5A1; displays >500-f..
RU-521 (RU.521, RU-320521) is a potent, selective cyclic GMP-AMP synthase (cGAS) inhibitor..
The first orally available, small-molecule TNIK inhibitor with IC50 of 21 nM; also weakly ..
ML241 is a potent, selective and reversible AAA ATPase p97 inhibitor (IC50=100 nM); blocks..
ML241 Hcl is a potent, selective and reversible AAA ATPase p97 inhibitor (IC50=100 nM); bl..
A potent, selective, allosteric and orally bioavailable protein tyrosine phosphatase SHP2 ..
SHP-099 (SHP099) is a potent, selective, allosteric and orally bioavailable protein tyrosi..
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