| Cat. No. |
Product Name |
Information |
| PC-36101 |
KH-176
ROS-redox modulator
|
KH-176 (KH176, Sonlicromanol) is a smal molecule ROS-redox modulator, effectively reduces increased cellular ROS levels and protects OXPHOS deficient primary cells against redox perturbation by targeting the Thioredoxin/Peroxiredoxin system. |
| PC-35973 |
MRS1186
A3AR antagonist
|
MRS1186 (MRS-1186) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist with Ki of 7.66 nM.. |
| PC-35841 |
AB928
A2AR/A2BR antagonist
|
Etrumadenant (AB928) is a potent, dual antagonist of the A2aR and A2bR adenosine receptors with Kb of 1.5 and 2.0 nM, respectively. |
| PC-35779 |
Taminadenant
A2AR antagonist
|
Taminadenant (PBF509, NIR178) is a novel selective and potent Adenosine A2A Receptor (A2AR) antagonist, antagonizes A2AR agonist-mediated cAMP accumulation and impedance responses with KB values of 72.8 and 8.2 nM, respectively. |
| PC-35507 |
MSX-3 hydrate
A2AR antagonist
|
MSX-3 hydrate is a potent, specific adenosine A2A receptor (A2AR) antagonist. |
| PC-35297 |
TP455
A2AR antagonist
|
TP455 (TP-455) is a highly potent, selective A2A adenosine receptor inverse agonist with IC50 of 1.9 nM in cyclic AMP assays in hA2A CHO cells. |
| PC-35002 |
BAY 60-6583
A2BR agonist
|
BAY 60-6583 (BAY60-6583) is a potent, selective adenosine A2B receptor (A2BR) agonist with EC50 of 2.83 nM (murine A2BR). |
| PC-63435 |
Neladenoson dalanate hydrochloride
A1AR agonist
|
Neladenoson dalanate (BAY 10-67197) is a potent, selective, orally acitve partial adenosine A1 receptor (A1AR) agonist (EC50=0.1 nM) for the treatment of chronic heart failure. |
| PC-63434 |
Neladenoson dalanate
A1AR agonist
|
Neladenoson dalanate (BAY 10-67197) is a potent, selective, orally acitve partial adenosine A1 receptor (A1AR) agonist (EC50=0.1 nM) for the treatment of chronic heart failure. |
| PC-43415 |
LUF6000
A3AR modulator
|
LUF6000 is a potent, selective, positive allosteric modulator (enhancer) of human A3 adenosine receptor, enhance Emax but without affecting agonist potency. |
| PC-43386 |
CGS21680 hydrochloride
A2AR agonist
|
CGS 21680 hydrochloride is a specific adenosine A2A subtype receptor agonist with Ki of 27 nM. |
| PC-43385 |
CGS21680
A2AAR agonist
|
CGS21680 is a potent, specific adenosine A2A subtype receptor agonist with Ki of 27 nM. |
