| Cat. No. |
Product Name |
Information |
| PC-45566 |
N6-Cyclohexyladenosine
A1AR agonist
|
N6-Cyclohexyladenosine is an adenosine A1 receptor agonist (EC50= 8.2 nM). |
| PC-44125 |
Capadenoson
A1AR agonist
|
Capadenoson (BAY68-4986) is a selective agonist of adenosine-A1 receptor (A1AR). |
| PC-42771 |
Tozadenant
A2AR antagonist
|
Tozadenant (SYN115) is a potent, selective adenosine 2A receptor (A2AR) antagonist with Ki of 11.5 nM. |
| PC-45585 |
GR-79236
A1AR agonist
|
GR-79236 is a potent and selective Adenosine A1 receptor agonist with Ki of 3.1 nM. |
| PC-42717 |
Vipadenant
A2AR antagonist
|
Vipadenant (BIIB014) is a potent and selective A2A adenosine receptor antagonist with Ki of 1.3 nM. |
| PC-42729 |
Preladenant
A2AR antagonist
|
Preladenant (SCH-420814, MK-3814) is a potent and highly selective adenosine A2A receptor competitive antagonist with Ki of 1.1 nM. |
| PC-42728 |
Istradefylline
A2AR antagonist
|
Istradefylline (KW-6002) is a potent and highly selective A2A receptor antagonist with Ki of 2.2 nM. |
| PC-45527 |
APNEA
A3AR agonist
|
APNEA is a non-selective agonist of adenosine A3 receptor, has a high affinity for the adenosine A1 and A3 receptors. |
| PC-45624 |
AB-MECA
A3AR agonist
|
AB-MECA is a high affinity A3 adenosine receptor (A3AR) agonist with binding Ki of 430.5 nM for human A3 receptors in CHO cells. |
| PC-25759 |
P626
A2AR/A2BR antagonist
|
P626 is a potent, selective dual adenosine A2A/A2B receptor (A2AR/A2BR) antagonist with IC50 of 5.73 nM and 34 nM at both hA2AAR and hA2BAR (cAMP assay), with no significant acitivity against hA1AR and hA3AR. |
| PC-25685 |
LJ-4378
A2AAR agonist, A3AR antagonist
|
LJ-4378 is a dual-acting ligand with A2AAR agonist (EC50=80.3 nM for cAMP formation, binding Ki=7.19 nM) and A3 adenosine receptor (A3AR, binding Ki=11.8 nM) antagonist activity. |
| PC-25476 |
MIPS2719
A1AR antagonist
|
MIPS2719 is a potent, selective, covalent, irreversible antagonist of A1 adenosine receptor (A1AR)with pKB value of 8.2, selective for the A1AR over the A2AAR. |
