| Cat. No. |
Product Name |
Information |
| PC-22021 |
Devazepide
CCK1 inhibitor
|
Devazepide (L-364,718) is a potent, competitive, selective and orally active nonpeptide antagonist of peripheral cholecystokinin (CCK) receptor with IC50 of 81 pM, 45 pM and 245 nM for rat pancreatic, bovine gallbladder and guinea pig brain CCK receptors. |
| PC-35949 |
SR146131
CCK1 inhibitor
|
SR146131 (SR-146131) a small molecule positive allosteric modulator of the type 1 cholecystokinin receptor (CCK1R) with pEC50 of 10.34. |
| PC-70239 |
L-365260
CCK2 inhibitor
|
L-365260 (L365260) is a potent, selective, orally active cholecystokinin receptor 2 (CCK2) antagonist with IC50 of 2 nM. |
| PC-70198 |
PF-04756956
CCK1 inhibitor
|
PF-04756956 is a potent, selective CCK1 receptor agonist with EC50 of 0.47 nM. |
| PC-70197 |
CE-326597
CCK1 agonist
|
CE-326597 is a potent, selective agonist of the human and rat CCK1 receptor with Ki of 36 nM. |
| PC-70196 |
JNJ-26070109
CCK2 inhibitor
|
JNJ-26070109 is a novel, potent, selective orally active CCK-2 receptor antagonist with pKi of 8.49 for hCCK2. |
| PC-60082 |
Netazepide
CCK2 inhibitor
|
Netazepide (YF476, Sograzepide) is a potent, selective and orally active gastrin/CCK-2 antagonist with IC50 of 0.1 nM. |
| PC-60036 |
Ceclazepide
CCK2 inhibitor
|
Ceclazepide is a potent, selective cholecystokinin receptor CCK2 antagonist for treatment of gastroesophageal reflux disease (GERD). |
| PC-45389 |
Z-360
CCK2 inhibitor
|
Z-360 (Nastorazepide) is a novel potent, orally active CCK-2/gastrin receptor antagonist with Ki of 0.47 nM. |
| PC-25772 |
CCKBR Gi-biased agonist 3qr
CCKBR agonist
|
CCKBR Gi-biased agonist 3qr is a potent, selective Gq-biased agonist of cholecystokinin (CCK) B receptor (CCKBR) with EC50 of 0.035 nM. |
| PC-25771 |
Lyz-866
CCKBR agonist
|
Lyz-866 is a potent, selective Gi-biased agonist of cholecystokinin (CCK) B receptor (CCKBR) with EC50 of 0.27 nM. |
| PC-25770 |
CCKBR agonist z-44
CCKBR agonist
|
CCKBR agonist z-44 is a potent, selective Gi-biased agonist of cholecystokinin (CCK) B receptor (CCKBR), does not activator CCKAR and Gq/Gs downstream signaling of CCKBR. |
