| Cat. No. |
Product Name |
Information |
| PC-60974 |
Gemigliptin
DPP-4 inhibitor
|
Gemigliptin (LC15-0444) is a potent, selective, competitive and orally active DPP4 inhibitor (IC50=10.4 nM, hDPP4) with potential for the treatment of type 2 diabetes. |
| PC-60517 |
Gosogliptin dihydrochloride
DPP-4 inhibitor
|
Gosogliptin dihydrochloride (PF-00734200) is a potent, selective, competitive, orally active dipeptidyl peptidase-4 (DPP-4) inhibitor with IC50 of 13 nM. |
| PC-60516 |
Gosogliptin
DPP-4 inhibitor
|
Gosogliptin (PF-734200, PF-00734200) is a potent, selective, competitive, orally active dipeptidyl peptidase-4 (DPP-4) inhibitor with IC50 of 13 nM. |
| PC-60515 |
Garvagliptin
DPP-4 inhibitor
|
Garvagliptin (NVP LAF 237A, LAF237A) is a potent, selective dipeptidyl peptidase-4 (DPP-4) inhibitor for treatment for type 2 diabetes. |
| PC-60297 |
AZD-7986
DPP-1 inhibitor
|
AZD-7986 (INS-1007, Brensocatib) is a highly potent, reversible, and selective DPP1 inhibitor with enzyme and cell pIC50 of 8.4. |
| PC-60064 |
Imigliptin dihydrochloride
DPP-4 inhibitor
|
Imigliptin dihydrochloride (KBP-3853) is a potent, selective, orally available DPP-4 inhibitor with IC50 of 9 nM. |
| PC-44866 |
Omarigliptin
DPP4 inhibitor
|
Omarigliptin (MK-3102) is a potent and selective DPP-4 inhibitor with IC50 of 1.4 nM. |
| PC-42224 |
SP-13786
FAP inhibitor
|
SP-13786 is a highly potent, selective, orally bioavailable inhibitor of fibroblast activation protein (FAP) with IC50 of 3.2 nM. |
| PC-42508 |
Linagliptin
DPP4 inhibitor
|
Linagliptin (BI-1356) is a highly potent, selective, long-acting, and orally bioavailable DPP-4 inhibitor with IC50 of 1 nM. |
| PC-42509 |
Saxagliptin
DPP4 inhibitor
|
Saxagliptin (BMS-477118) is a highly potent, long-acting, orally active DPP4 inhibitor with Ki of 0.6 nM. |
| PC-20822 |
Nateglinide
DPP IV inhibitor
|
Nateglinide (Senaglinide, DJN-608, A-4166) is an oral hypoglycaemic agent and non-sulphonylurea insulin secretagogue, also is a MRGPRX4 agonist. |
| PC-20348 |
Sitagliptin phosphate
DPP-4 inhibitor
|
Sitagliptin phosphate (MK-0431, MK0431) is a potent, orally active dipeptidyl peptidase IV (DPP4) inhibitor with IC50 of 18 nM. |
