| Cat. No. |
Product Name |
Information |
| PC-72083 |
FPR1 agonist fMLF
FPR1 agonist
|
FPR1 agonist fMLF (NSC 350593) is a potent, selective formylpeptide receptor-1 (FPR1) agonist with EC50 of 80 nM in calcium flux, Ki of 38 nM. |
| PC-72082 |
ICT12035
FPR1 antagonist
|
ICT12035 (AZ2158) is a potent, selective formylpeptide receptor-1 (FPR1) antagonist with IC50 of 30 nM in calcium mobilisation assays (100 nM fMLF). |
| PC-62594 |
ACT-389949
FPR2 agonist
|
ACT-389949 (ACT389949) is a novel potent and selective formyl peptide receptor type 2 (FPR2)/Lipoxin A4 receptor (ALX) agonist with EC50 of 3 nM for FPR2/ALX internalization into monocytes. |
| PC-26925 |
Boc-MLF TFA
FPR1 antagonist
|
Boc-MLF TFA (Boc-1, Boc-Met-Leu-Phe-OH) is a specific, peptide FPR1 antagonist, reduces superoxide production induced by fMLF with IC50 of 0.63 uM. |
| PC-26924 |
Boc-MLF
FPR1 antagonist
|
Boc-MLF (Boc-1, Boc-Met-Leu-Phe-OH) is a specific, peptide FPR1 antagonist, reduces superoxide production induced by fMLF with IC50 of 0.63 uM. |
| PC-26923 |
fMLFC
FPR1 agonist
|
fMLFC (fMet-Leu-Phe-Cys) is a peptide agonist of formyl peptide receptor 1 (FPR1), induces lysosomal degradation of FPR1, effectively reduces cell surface FPR1 expression by preventing its recycling after endocytosis, ameliorates lung injury in LPS-treated mice. |
| PC-26270 |
BMS-986331
FPR2 agonist
|
BMS-986331 is a highly potent and selective Formyl peptide receptor 2 (FPR2) agonist with EC50 of 0.5 nM (hFPR2). |
| PC-25276 |
N-19004
FPR1 antagonist
|
N-19004 is a potent, specific formyl peptide receptor (FPR1) antagonist with IC50 of 68.9 nM for inhibition of the binding of FITC-fMLF to THP-1 cells. |
| PC-24177 |
FPR2 agonist compound 8
FPR2 agonist
|
FPR2 agonist compound 8 is a potent, selective agonist of formyl peptide receptor 2 (FPR2/ALX, Lipoxin A4 Receptor) with β-arrestin recruitment EC50 of 20 nM, calcium mobilization EC50 of 740 nM. |
