| Cat. No. |
Product Name |
Information |
| PC-49655 |
PSB-0952
CD73 inhibitor
|
PSB-0952 (PSB0952) is a potent, selective ecto-5'-Nucleotidase (eN, CD73) inhibitor with Ki of 260 nM, >150-fold selectivity over NTPDases and P2Y receptor subtypes P2Y2, P2Y4, P2Y6, and P2Y12. |
| PC-49654 |
PSB-0963
CD73 inhibitor
|
PSB-0963 (PSB0963) is a potent, selective ecto-5'-Nucleotidase (eN, CD73) inhibitor with Ki of 150 nM, >100-fold selectivity over NTPDases. |
| PC-49421 |
Oroxylin A
Transketolase inhibitor
|
Oroxylin A is a small molecule transketolase (TKT) inhibitor with SPR KD of 70.7 uM, inhibits hepatocellular carcinoma growth in vitro and in vivo. |
| PC-38899 |
TAS1553
RNR inhibitor
|
TAS1553 is a highly potent, selective small-molecule inhibitor of ribonucleotide reductase (RNR) with enzyme IC50 of 54.2 nM, binds to R1 subunit with Kd of 34.9 nM, disrupts PPI between R1 and R2 subunit. |
| PC-38835 |
DI-87
dCK inhibitor
|
DI-87 ((R)-DI-87) is a highly potent, specific, orally bioavailable deoxycytidine kinase (dCK) inhibitor with IC50 of 3.15 nM. |
| PC-38579 |
3-Deazauridine
CTP inhibitor
|
3-Deazauridine (DAU, NSC 126849) is a nucleoside analog that competitively inhibits cytidine triphosphate synthetase (CTP). |
| PC-38453 |
YMU1
hTMPK inhibitor
|
YMU1 is a specific, cell-permeable inhibitor of human thymidylate kinase (hTMPK) with IC50 of 0.61 uM in enzymatic assays. |
| PC-72499 |
N6-benzyladenosine
DNPH1 inhibitor
|
N6-benzyladenosine (DNPH1i, N6-benzyl-AMP) is a nucleoside analog that acts as competitive inhibitor of deoxynucleotide N-hydrolase DNPH1. |
| PC-72483 |
MRT00252040
PAICS inhibitor
|
MRT00252040 (PAICSi) is a small molecule inhibitor PAICS, which catalyzes two steps in the de novo purine synthesis pathway. |
| PC-36085 |
Aspacytarabine
|
Aspacytarabine (Astarabine, BST236) is a cytarabine conjugate that shows anti-neoplastic agents for inhibiting cancer cell growth. . |
| PC-35966 |
Thymidine Phosphorylase inhibitor TPI
|
Thymidine Phosphorylase inhibitor TPI (hTP inhibitor TPI) is a potent, selective inhibitor of thymidine phosphorylase (TPase) with Ki of 17 nM, does not inhibits uridine phosphorylase, thymidine kinase, orotate phosphoribosyltransferase, or dihydropyrimidine dehydrogenase. |
| PC-35560 |
Elacytarabine
|
Elacytarabine (CP-4055, CP4055, ELACYT) is a fatty acid derivative of cytarabine with potential antineoplastic activity. |
