| Cat. No. |
Product Name |
Information |
| PC-35539 |
NFEPP
|
NFEPP is a novel potent, selective pH-dependent μ-opioid receptor (MOR) agonist with a low pKa, shows significantly lower affinity compared with fentanyl at pH 7.4. |
| PC-43173 |
Nalfurafine hydrochloride
|
Nalfurafine (TRK-820, TRK820) is potent, selective agonist of kappa-opioid receptor with Ki of 3.5 nM, 15-fold less potent for μOR and little affinity for δOR (Ki=53 and 1,200 nM, respectively). |
| PC-43172 |
Nalfurafine
|
Nalfurafine (TRK-820, TRK820) is potent, selective agonist of kappa-opioid receptor with Ki of 3.5 nM, 15-fold less potent for μOR and little affinity for δOR (Ki=53 and 1,200 nM, respectively). |
| PC-42356 |
PZM21
|
PZM21 is a potent, selective Gi-biased μ-opioid-receptor (μOR) agonist with Ki/EC50 of 1.1/4.6 nM, has little to no detectable κOR/δOR agonist or nociceptin receptor agonist activity. |
| PC-62111 |
ML350
|
ML350 (CYM 50202) is a highly potent and selective Opioid kappa receptor (OPRK1/KOR) antagonist with IC50 of 9-16 nM. |
| PC-62109 |
PF-04455242 hydrochloride
|
PF-04455242 is a potent, selective κ-opioid receptor (KOR) antagonist with Ki of 3 nM/21 nM/22 nM for hKOR/rKOR/mKOR, respectively. |
| PC-62108 |
PF-04455242
|
PF-04455242 is a potent, selective κ-opioid receptor (KOR) antagonist with Ki of 3 nM/21 nM/22 nM for hKOR/rKOR/mKOR, respectively. |
| PC-62107 |
Enadoline
|
Enadoline (CI 977. |
| PC-61887 |
Spiradoline mesylate
|
Spiradoline (U 62066) is a potent, highly selective κ-opioid agonist that has analgesic diuretic and antitussive effects.. |
| PC-61886 |
Spiradoline
|
Spiradoline (U 62066) is a potent, highly selective κ-opioid agonist that has analgesic diuretic and antitussive effects.. |
| PC-61596 |
SR-8993
|
A potent, highly selective, brain-penetrant NOP-R (Nociceptin/orphanin FQ receptor) agonist with EC50 of 8.8 nM. |
| PC-61550 |
AT-127
|
AT-127 is a novel potent, selective nociceptin/orphanin FQ receptor (NOP receptor) agonist with Ki of 1.18 nM. |
