| Cat. No. |
Product Name |
Information |
| PC-21615 |
SRX-246
V1a receptor antagonist
|
SRX-246 (SRX246) is a potent, selective and CNS penetrant human V1a receptor antagonist with Ki of 0.3 nM. |
| PC-21614 |
RGH-122
V1a receptor antagonist
|
RGH-122 is a potent, selective, and orally bioavailable V1a receptor antagonist with Ki/IC50 of 0.3/0.9 nM (hV1a) respectively, >100-fold selectiive over V2 receptor. |
| PC-21436 |
SR-49059
V1AR antagonist
|
SR49059 (SR-49059) is a potent, selective and orally active vasopressin V1a antagonist with Ki of 1.4 nM. |
| PC-49652 |
OPC-61815
V2R inhibitor
|
OPC-61815 is a water-soluble phosphate ester pro-drug of Tolvaptan (Cat# PC-45125), which is an orally active vasopressin V2 receptor antagonist. |
| PC-38647 |
Enuvaptan
V1AR antagonist
|
Enuvaptan (BAY2327949) is a potent, selective vasopressin 1a receptor (V1AR) antagonist with potential for renal and cardiovascular diseases. |
| PC-62116 |
ML389
|
ML389 is a highly potent, selective vasopressin receptor 1a (V1a-R) antagonist with IC50 of 40 nM. |
| PC-61507 |
TASP0434299
|
A radioligand candidate for arginine vasopressin 1B (V1B) receptor that exhibits high binding affinities for human and rat V1B receptors with IC50 of 0.526 and 0.641 nM, respectively. |
