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Cat. No. Product Name Information
PC-73282

DC-TEADin1072

TEAD1/3 inhibitor

DC-TEADin1072 is a novel TEAD1/3 covalent inhibitor with biochemical IC50 values of 0.61 and 0.58 uM against TEAD1 and TEAD3, respectively.
PC-72427

LM98

YAP-TEAD inhibitor

LM98 (TEAD inhibitor LM98) is a flufenamic acid analogue, shows strong affinity to TEAD, inhibits its autopalmitoylation and reduces the YAP-TEAD transcriptional activity.

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