| Cat. No. |
Product Name |
Information |
| PC-60764 |
A 834735
Cannabinoid receptor agonist
|
A 834735 is a potent, nonselective, brain penetrant, full agonist at both the central CB1 and peripheral CB2 receptors with Ki of 4.6 and 0.31 nM, respectively. |
| PC-60763 |
JTE907
CB2 inverse agonist
|
JTE907 (JTE-907) is a potent, selective, orally active cannabinoid CB2 receptor inverse agonist with Ki of 35.9, 1.55 and 0.38 nM for human, mouse and rat CB2, respectively. |
| PC-60762 |
UR-144
CB2 agonist
|
UR-144 is a potent, selective full agonist of the peripheral cannabinoid receptor CB2 with Ki of 1.8 nM, >80-fold selectivity over CB1 (Ki=150 nM). |
| PC-60761 |
AM-2201
Cannabinoid receptor agonist
|
AM-2201 is a synthetic cannabinoid that acts as a potent, nonselective full agonist for the cannabinoid receptor with EC50 of 38 and 58 nM for CB1 and CB2, respectively. |
| PC-60760 |
AM-630
CB2 inverse agonist
|
AM-630 (6-Iodopravodoline) is a potent and selective inverse agonist for the cannabinoid receptor CB2 with Ki of 32.1 nM, 165-fold selectivity over CB1. |
| PC-60759 |
AM-1221
CB1 agonist
|
AM-1221 is a potent and selective agonist for the cannabinoid receptor CB1 with Ki of 0.28 nM, 180-fold selectivity over CB2. |
| PC-60758 |
MN-25
CB2 agonist
|
CB2 agonist MN25 (AR12) is a potent, reasonably selective agonist of peripheral cannabinoid receptor with Ki of 11 nM for CB2, 22-fold selectivity over the psychoactive CB1 receptors (Ki=245 nM). |
| PC-60757 |
NESS-0327
CB1R antagonist
|
NESS-0327 (NESS0327) is a potent, selective CB1 cannabinoid receptor antagonist with Ki of 350 fM, >60,000-fold selective for the CB1 receptor versus CB2 receptor (Ki=21 nM). |
| PC-60756 |
NESS-040C5
CB2 agonist
|
A potent, reasonably selective cannabinoid CB2 agonist with Ki of 0.4 nM, 25-fold selectivity over CB1 receptor.. |
| PC-60753 |
SR 144528
CB2 antagonist
|
SR 144528 is a highly potent, selective and orally active antagonist of CB2 receptor with Ki of 0.6 nM. |
| PC-60729 |
AM1241
CB2 agonist
|
AM1241 is a potent, selective cannabinoid receptor CB2 agonist with Ki of 7.1 nM, >80-fold selectivity over CB1 receptors in radioligand binding assay. |
| PC-60728 |
GW405833 hydrochloride
CB2 agonist
|
GW405833 is a potent, selective cannabinoid receptor CB2 agonist with Ki of 3.6 nM, 1200-fold selectivity over CB1. |
