| Cat. No. |
Product Name |
Information |
| PC-42171 |
Bay 59-3074
CB1/CB2 agonist
|
Bay 59-3074 is a potent, selective cannabinoid CB1/CB2 receptor partial agonist with Ki of 48.3, and 45.5 nM for human CB1 and human CB2 receptors, respectively. |
| PC-42063 |
Taranabant
CB1 inverse agonist
|
Taranabant (MK-0364) is a potent, selective and orally active cannabinoid-1 receptor (CB1R) inverse agonist with IC50 of 2.8 nM, Ki of 0.13 nM. |
| PC-42723 |
Otenabant
CB1 antagonist
|
Otenabant (CP-945598) is a potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively. |
| PC-27963 |
LEI-101
CB2R agonist
|
LEI-101 (LEI 101) is a potent, selective, orally available and peripherally restricted cannabinoid CB2 receptor agonist with binding pKi of 7.5 (hCB2R). |
| PC-27323 |
PM289
CB2R agonist
|
PM289 is a high affinity, selective Cannabinoid 2 Receptor (CB2R) agonist with Ki of 92.6 nM (hCB2), >300-fold selectivity over hCB1 receptors. |
| PC-26853 |
CP-55940
CB1R agonist
|
CP-55940 (CP55940) is a potent, selective cannabinoid receptor 1 (CB1R) agonist. |
| PC-26472 |
GW833972A
BMAL2 inhibitor, CB2 agonist
|
GW833972A is a potent, selective CB2 receptor agonist with pEC50 of 7.3 and 7.5 for human and rat CB2 receptors respecitvely, shows 1000-fold selectivity over CB1 receptor, also binds BMAL2 with high affinity and facilitates its protein degradation. |
| PC-26303 |
AM11101
CB1 receptor agonist
|
AM11101 is a potent cannabinoid CB1 receptor agonist with Ki /EC50 of 0.9/4.4 nM (rCB1), increases food intake in female rats. |
| PC-26033 |
A-796260
CB2 agonist
|
A-796260 is a potent, selective cannabinoid CB2 receptor agonist with binding Ki of 4.37 nM and 13.0 nM for human and rat CB2 receptors respectively, >30-fold selective over CB1 receptor. |
| PC-26032 |
PF-03550096
CB2 agonist
|
PF-03550096 is a potent, selective orally active cannabinoid receptor 2 (CB2) agonist with Ki of 7.9 nM and 47 nM for human and rat CB2 receptors respectively. |
| PC-26031 |
MDA77
CB2 inverse agonist
|
MDA77 is a potent selective cannabinoid receptor 2 (CB2) inverse agonist with EC50 of 5.82 nM at human CB2, with no activity at CB1, inhibits the effect of MDA7 (CB2 agonist) in animal model of neuropathic pain. |
| PC-26030 |
GW842166X
CB2 agonist
|
GW842166X (GW-842,166X) is a potent and selective cannabinoid receptor 2 (CB2) agonist with IC50 of 63 and 91 nM for human and rat CB2, respectively. |
