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Request The Product List ofCannabinoid Receptor Cannabinoid Receptor

Cat. No. Product Name Information
PC-60762

UR-144

A potent, selective full agonist of the peripheral cannabinoid receptor CB2 with Ki of 1.8 nM, >80-fold selectivity over CB2 (Ki=150 nM).
PC-60759

AM-1221

A potent and selective agonist for the cannabinoid receptor CB1 with Ki of 0.28 nM, 180-fold selectivity over CB2..
PC-60758

MN-25

A potent, reasonably selective agonist of peripheral cannabinoid receptor with Ki of 11 nM for CB2, 22-fold selectivity over the psychoactive CB1 receptors (Ki=245 nM)..
PC-60757

NESS-0327

A potent, selective CB1 cannabinoid receptor antagonist with Ki of 350 fM, >60,000-fold selective for the CB1 receptor versus CB2 receptor (Ki=21 nM).
PC-60756

NESS-040C5

A potent, reasonably selective cannabinoid CB2 agonist with Ki of 0.4 nM, 25-fold selectivity over CB1 receptor..
PC-60753

SR 144528

A highly potent, selective and orally active antagonist of CB2 receptor with Ki of 0.6 nM.
PC-60729

AM1241

A potent, selective cannabinoid receptor CB2 agonist with Ki of 7.1 nM, >80-fold selectivity over CB1 receptors in radioligand binding assay.
PC-60728

GW405833 hydrochloride

A potent, selective cannabinoid receptor CB2 agonist with Ki of 3.6 nM, 1200-fold selectivity over CB1.
PC-45531

JD-5037

A selective, peripherally restricted cannabinoid-1(CB1) receptor blocker with IC50 of 1.5 nM.
PC-42063

Taranabant

A potent, selective and orally active cannabinoid-1 receptor (CB1R) inverse agonist with IC50 of 2.8 nM, Ki of 0.13 nM.
PC-42724

Otenabant hydrochloride

A potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively.
PC-42723

Otenabant

A potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively.

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