Cat. No. |
Product Name |
Information |
PC-60762 |
UR-144
|
A potent, selective full agonist of the peripheral cannabinoid receptor CB2 with Ki of 1.8 nM, >80-fold selectivity over CB2 (Ki=150 nM). |
PC-60759 |
AM-1221
|
A potent and selective agonist for the cannabinoid receptor CB1 with Ki of 0.28 nM, 180-fold selectivity over CB2.. |
PC-60758 |
MN-25
|
A potent, reasonably selective agonist of peripheral cannabinoid receptor with Ki of 11 nM for CB2, 22-fold selectivity over the psychoactive CB1 receptors (Ki=245 nM).. |
PC-60757 |
NESS-0327
|
A potent, selective CB1 cannabinoid receptor antagonist with Ki of 350 fM, >60,000-fold selective for the CB1 receptor versus CB2 receptor (Ki=21 nM). |
PC-60756 |
NESS-040C5
|
A potent, reasonably selective cannabinoid CB2 agonist with Ki of 0.4 nM, 25-fold selectivity over CB1 receptor.. |
PC-60753 |
SR 144528
|
A highly potent, selective and orally active antagonist of CB2 receptor with Ki of 0.6 nM. |
PC-60729 |
AM1241
|
A potent, selective cannabinoid receptor CB2 agonist with Ki of 7.1 nM, >80-fold selectivity over CB1 receptors in radioligand binding assay. |
PC-60728 |
GW405833 hydrochloride
|
A potent, selective cannabinoid receptor CB2 agonist with Ki of 3.6 nM, 1200-fold selectivity over CB1. |
PC-45531 |
JD-5037
|
A selective, peripherally restricted cannabinoid-1(CB1) receptor blocker with IC50 of 1.5 nM. |
PC-42063 |
Taranabant
|
A potent, selective and orally active cannabinoid-1 receptor (CB1R) inverse agonist with IC50 of 2.8 nM, Ki of 0.13 nM. |
PC-42724 |
Otenabant hydrochloride
|
A potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively. |
PC-42723 |
Otenabant
|
A potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively. |