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Cat. No. Product Name Information
PC-35435

UniPR1331

Eph-ephrin inhibitor

UniPR1331 (UniPR-1331) is a selective, orally available antagonist of Eph/ephrin interaction with pIC50 of 5.45, IC50 of 2.9 uM.
PC-43438

NVP-BHG712

EphB4 inhibitor

NVP-BHG712 is a potent, specific inhibitor of EphB4 kinase that inhibits EphB4 autophosphorylation with IC50 of 25 nM in cell-bases assays, displays little to no activity against VEGFR2, IGF1R and InsR.
PC-45397

ALW-II-41-27

EPHA2 inhibitor

ALW-II-41-27 is an ATP-competitive EPHA2 RTK inhibitor with IC50 of 11 nM.
PC-21784

WCDD301

EphA4 agonist

WCDD301 is a high-affinity, orally available agonist of EphA4 receptor.
PC-20805

UniPR129

Ephrin Receptor antagonist

UniPR129 is a potent, selective Eph/ephrin antagonist, competitively disrupts Eph2A-ephrin-A1 binding (IC50=945 nM, Ki = 345 nM).
PC-49438

Targefrin

EphA2-LBD inhibitor

Targefrin is a potent, selective antagonist targeting ligand binding domain of receptor tyrosine kinase EphA2 (EphA2-LBD), binds to EphA2-LBD with Kd of 21 nM (ITC) and shows IC50 value of 10.8 nM in biochemical assays.
PC-62858

EphB3-IN-1

EphB3-IN-1 is the first potent, selective inhibitor of EphB3 that exhibits inhibiting EphB3 autophosphorylation in cells with IC50 of 3 nM.

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